Tuning the properties of penetrating peptides by oxime conjugation

We here describe the application of oxime bond formation between a peptide scaffold and different aldehydes to modify the transporting capabilities of penetrating peptides. We show that bonds such as oximes offer a great synthetic advantage for the modification of the properties of model penetrating...

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Detalhes bibliográficos
Autores: Pazo Pascual, Marta, Fernández Caro, Héctor, Priegue Caamaño, Juan Manuel, Lostalé Seijo, Irene, Montenegro García, Javier
Tipo de documento: artigo
Data de publicação:2017
País:España
Recursos:Universidad de Santiago de Compostela (USC)
Repositório:Minerva. Repositorio Institucional de la Universidad de Santiago de Compostela
Idioma:inglês
OAI Identifier:oai:minerva.usc.gal:10347/15141
Acesso em linha:http://hdl.handle.net/10347/15141
Access Level:Acceso aberto
Palavra-chave:Materias::Investigación::23 Química::2302 Bioquímica
Descrição
Resumo:We here describe the application of oxime bond formation between a peptide scaffold and different aldehydes to modify the transporting capabilities of penetrating peptides. We show that bonds such as oximes offer a great synthetic advantage for the modification of the properties of model penetrating peptides. We believe that this approach will allow the development of improved intracellular delivery vehicles