Pharmacognostic evaluation of Libidibia ferrea extracts and analysis of semi-solid dosage forms

A medicinal plant known as Jucá (Libidibia ferrea) is a Brazilian tree that possesses several therapeutic uses, including wound healing actions, due to the presence of polyphenols. Fruits from Libidibia ferrea var. leiostachya (Benth.) L.P. and Libidibia ferrea (Mart. ex Tul.) L.P. Queiroz var. ferr...

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Autores: Morel, Lucas Junqueira de Freitas, Nascimento Júnior, José Elvino do, França, Suzelei de Castro, Dandaro, Ivanice Maria Cestari, Borella , Júlio Cézar, Pereira, Ana Maria Soares
Formato: artículo
Estado:Versión publicada
Fecha de publicación:2023
País:Brasil
Recursos:Fundação Oswaldo Cruz (FIOCRUZ)
Repositorio:Revista Fitos
Idioma:inglés
OAI Identifier:oai:ojs.revistafitos.far.fiocruz.br:article/1492
Acesso em linha:https://revistafitos.far.fiocruz.br/index.php/revista-fitos/article/view/1492
Access Level:acceso abierto
Palavra-chave:Libidibia ferrea
Brazilian Ironwood
Production of Herbal Medicines
Quality control
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dc.title.none.fl_str_mv Pharmacognostic evaluation of Libidibia ferrea extracts and analysis of semi-solid dosage forms
Avaliação farmacognóstica de extratos de Libidibia ferrea e análise de formas farmacêuticas semissólidas.
title Pharmacognostic evaluation of Libidibia ferrea extracts and analysis of semi-solid dosage forms
spellingShingle Pharmacognostic evaluation of Libidibia ferrea extracts and analysis of semi-solid dosage forms
Morel, Lucas Junqueira de Freitas
Libidibia ferrea
Brazilian Ironwood
Production of Herbal Medicines
Quality control
title_short Pharmacognostic evaluation of Libidibia ferrea extracts and analysis of semi-solid dosage forms
title_full Pharmacognostic evaluation of Libidibia ferrea extracts and analysis of semi-solid dosage forms
title_fullStr Pharmacognostic evaluation of Libidibia ferrea extracts and analysis of semi-solid dosage forms
title_full_unstemmed Pharmacognostic evaluation of Libidibia ferrea extracts and analysis of semi-solid dosage forms
title_sort Pharmacognostic evaluation of Libidibia ferrea extracts and analysis of semi-solid dosage forms
dc.creator.none.fl_str_mv Morel, Lucas Junqueira de Freitas
Nascimento Júnior, José Elvino do
França, Suzelei de Castro
Dandaro, Ivanice Maria Cestari
Borella , Júlio Cézar
Pereira, Ana Maria Soares
author Morel, Lucas Junqueira de Freitas
author_facet Morel, Lucas Junqueira de Freitas
Nascimento Júnior, José Elvino do
França, Suzelei de Castro
Dandaro, Ivanice Maria Cestari
Borella , Júlio Cézar
Pereira, Ana Maria Soares
author_role author
author2 Nascimento Júnior, José Elvino do
França, Suzelei de Castro
Dandaro, Ivanice Maria Cestari
Borella , Júlio Cézar
Pereira, Ana Maria Soares
author2_role author
author
author
author
author
dc.subject.por.fl_str_mv Libidibia ferrea
Brazilian Ironwood
Production of Herbal Medicines
Quality control
topic Libidibia ferrea
Brazilian Ironwood
Production of Herbal Medicines
Quality control
description A medicinal plant known as Jucá (Libidibia ferrea) is a Brazilian tree that possesses several therapeutic uses, including wound healing actions, due to the presence of polyphenols. Fruits from Libidibia ferrea var. leiostachya (Benth.) L.P. and Libidibia ferrea (Mart. ex Tul.) L.P. Queiroz var. ferrea, were collected in Teresina (PI) and Jardinópolis (SP), respectively, and were used to prepare hydroethanolic and hydroglycolic extracts, produced in a 1:10 ratio. The extracts from the fruits from L. ferrea var. ferrea were used for the preparation of creams and ointments, containing 10 % (w/w) of these extracts. The extracts prepared with the fruits from L. ferrea var. ferrea (PI) are twice as concentrated in gallic acid content and in the percentage of dry residue, in comparison with those obtained from the fruits L. ferrea var. leiostachya. Among the formulations prepared, creams and ointments showed, statistically, the same concentration of total phenols, regardless of the type of extract used. The spreadability evaluation, which refers to the distribution of the pharmaceutical form by application area, showed that creams and ointments had very similar behaviors, except for the ointment produced with hydroglycolic extract, which was very fluid, making its therapeutic use unfeasible.
publishDate 2023
dc.date.none.fl_str_mv 2023-12-20
dc.type.driver.fl_str_mv info:eu-repo/semantics/article
info:eu-repo/semantics/publishedVersion
format article
status_str publishedVersion
dc.identifier.uri.fl_str_mv https://revistafitos.far.fiocruz.br/index.php/revista-fitos/article/view/1492
10.32712/2446-4775.2023.1492
url https://revistafitos.far.fiocruz.br/index.php/revista-fitos/article/view/1492
identifier_str_mv 10.32712/2446-4775.2023.1492
dc.language.iso.fl_str_mv eng
language eng
dc.relation.none.fl_str_mv https://revistafitos.far.fiocruz.br/index.php/revista-fitos/article/view/1492/1417
https://revistafitos.far.fiocruz.br/index.php/revista-fitos/article/view/1492/1412
dc.rights.driver.fl_str_mv Copyright (c) 2023 Revista Fitos
https://creativecommons.org/licenses/by/4.0
info:eu-repo/semantics/openAccess
rights_invalid_str_mv Copyright (c) 2023 Revista Fitos
https://creativecommons.org/licenses/by/4.0
eu_rights_str_mv openAccess
dc.format.none.fl_str_mv application/pdf
text/html
dc.publisher.none.fl_str_mv Centro de Inovação em Biodiversidade e Saúde - Farmanguinhos/Fiocruz
publisher.none.fl_str_mv Centro de Inovação em Biodiversidade e Saúde - Farmanguinhos/Fiocruz
dc.source.none.fl_str_mv Revista Fitos; Vol. 17 No. 4 (2023); 513-527
Revista Fitos; Vol. 17 Núm. 4 (2023); 513-527
Revista Fitos; v. 17 n. 4 (2023); 513-527
2446-4775
1808-9569
reponame:Revista Fitos
instname:Fundação Oswaldo Cruz (FIOCRUZ)
instacron:FIOCRUZ
instname_str Fundação Oswaldo Cruz (FIOCRUZ)
instacron_str FIOCRUZ
institution FIOCRUZ
reponame_str Revista Fitos
collection Revista Fitos
repository.name.fl_str_mv Revista Fitos - Fundação Oswaldo Cruz (FIOCRUZ)
repository.mail.fl_str_mv revistafitos@far.fiocruz.br || eugenio.telles@far.fiocruz.br
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spelling Pharmacognostic evaluation of Libidibia ferrea extracts and analysis of semi-solid dosage formsAvaliação farmacognóstica de extratos de Libidibia ferrea e análise de formas farmacêuticas semissólidas. Libidibia ferreaBrazilian IronwoodProduction of Herbal MedicinesQuality controlA medicinal plant known as Jucá (Libidibia ferrea) is a Brazilian tree that possesses several therapeutic uses, including wound healing actions, due to the presence of polyphenols. Fruits from Libidibia ferrea var. leiostachya (Benth.) L.P. and Libidibia ferrea (Mart. ex Tul.) L.P. Queiroz var. ferrea, were collected in Teresina (PI) and Jardinópolis (SP), respectively, and were used to prepare hydroethanolic and hydroglycolic extracts, produced in a 1:10 ratio. The extracts from the fruits from L. ferrea var. ferrea were used for the preparation of creams and ointments, containing 10 % (w/w) of these extracts. The extracts prepared with the fruits from L. ferrea var. ferrea (PI) are twice as concentrated in gallic acid content and in the percentage of dry residue, in comparison with those obtained from the fruits L. ferrea var. leiostachya. Among the formulations prepared, creams and ointments showed, statistically, the same concentration of total phenols, regardless of the type of extract used. The spreadability evaluation, which refers to the distribution of the pharmaceutical form by application area, showed that creams and ointments had very similar behaviors, except for the ointment produced with hydroglycolic extract, which was very fluid, making its therapeutic use unfeasible.A planta medicinal conhecida como Jucá (Libidibia ferrea) é uma árvore brasileira que possui diversos usos terapêuticos, incluindo ação cicatrizante, devido à presença de polifenóis. Libidibia ferrea var. leiostachya (Benth.) L.P. e Libidibia ferrea (Mart. ex Tul.) L.P. Queiroz var. ferrea, foram coletados em Teresina (PI) e Jardinópolis (SP), respectivamente, e foram utilizados para preparar extratos hidroetanólico e hidroglicólico, produzidos na proporção 1:10. Extratos dos frutos de L. ferrea var. ferrea foram utilizados para a preparação de cremes e pomadas, contendo 10% (p/p) desses extratos. Extratos preparados com os frutos de L. ferrea var. ferrea (PI) são duas vezes mais concentrados no teor de ácido gálico e na porcentagem de resíduo seco, em comparação com os obtidos a partir de frutos L. ferrea var. leiostachya. Entre as formulações elaboradas, os cremes e pomadas apresentaram estatisticamente a mesma concentração de fenóis totais, independente do tipo de extrato utilizado. A avaliação da espalhabilidade, que se refere à distribuição da forma farmacêutica por área de aplicação, mostrou que cremes e pomadas tiveram comportamentos muito semelhantes, com exceção da pomada produzida com extrato hidroglicólico, que se mostrou bastante fluida, tornando seu uso terapêutico inviável.Centro de Inovação em Biodiversidade e Saúde - Farmanguinhos/Fiocruz2023-12-20info:eu-repo/semantics/articleinfo:eu-repo/semantics/publishedVersionapplication/pdftext/htmlhttps://revistafitos.far.fiocruz.br/index.php/revista-fitos/article/view/149210.32712/2446-4775.2023.1492Revista Fitos; Vol. 17 No. 4 (2023); 513-527Revista Fitos; Vol. 17 Núm. 4 (2023); 513-527Revista Fitos; v. 17 n. 4 (2023); 513-5272446-47751808-9569reponame:Revista Fitosinstname:Fundação Oswaldo Cruz (FIOCRUZ)instacron:FIOCRUZenghttps://revistafitos.far.fiocruz.br/index.php/revista-fitos/article/view/1492/1417https://revistafitos.far.fiocruz.br/index.php/revista-fitos/article/view/1492/1412Copyright (c) 2023 Revista Fitoshttps://creativecommons.org/licenses/by/4.0info:eu-repo/semantics/openAccess Morel, Lucas Junqueira de FreitasNascimento Júnior, José Elvino doFrança, Suzelei de CastroDandaro, Ivanice Maria CestariBorella , Júlio CézarPereira, Ana Maria Soares2024-01-24T15:18:42Zoai:ojs.revistafitos.far.fiocruz.br:article/1492Revistahttps://revistafitos.far.fiocruz.br/index.php/revista-fitos/PUBhttp://revistafitos.far.fiocruz.br/index.php/revista-fitos/oairevistafitos@far.fiocruz.br || eugenio.telles@far.fiocruz.br2446-47752446-4775opendoar:2024-01-24T15:18:42Revista Fitos - Fundação Oswaldo Cruz (FIOCRUZ)false
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